GABAA receptor agent 2 TFA
GABAA receptor agent 2 TFA is a potent and selective GABAA receptor antagonist, exhibiting high affinity with an IC50 of 24 nM at human α1β2γ2 receptors and a Ki of 28 nM at rat receptors. It shows no activity against human GABA transporters (hGAT-1, hBGT-1, hGAT-2, hGAT-3), making it a useful tool for studying GABAergic neurotransmission in neuropharmacology and electrophysiology research.
Product Specifications
CAS Number
1781880-44-1
Field of Research
Neuroscience, Neuroscience; Immunology & Inflammation, Pharmacology & Drug Discovery
Smiles
O=C (O) C (F) (F) F.ON1N=CC (=C1C=2C=CC=C (C2) C=3C=CC=CC3) C4CCNCC4
Molecular Formula
C22H22F3N3O3
Molecular Weight
433.42
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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