HIV-1 inhibitor-40
HIV-1 inhibitor-40 (Compound 4ab) is a potent non-nucleoside reverse transcriptase inhibitor (NNRTI) with an EC50 of 1.9 nM. It demonstrates in vivo efficacy against HIV-1 replication without significant acute toxicity, though it also acts as a sensitive CYP inhibitor via orexin receptor antagonism, a consideration for drug interaction studies.
Product Specifications
Field of Research
Infectious Disease & Virology, Infectious Disease & Virology; Pharmacology & Drug Discovery, Metabolism Research, Protein Biochemistry
Molecular Formula
C25H18N6O2
Molecular Weight
434.45
Storage Conditions
-20°C
Notes
For research use only.
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