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TRPC5-IN-4

TRPC5-IN-4 is a potent and selective TRPC5/TRPC4 inhibitor with IC50 values of 14.07 nM and 65 nM, respectively. It demonstrates a favorable safety profile with no observed hepatotoxicity or nephrotoxicity, supporting its use in research models for chronic kidney disease and related cardiovascular pathologies.

Product Specifications

CAS Number

2762315-39-7

Field of Research

Pharmacology & Drug Discovery, Signal Transduction

Smiles

O (C1=C2C (CN (CC2) C3=C (Cl) C (=O) NC3=O) =NC=N1) C4=C (C (F) (F) F) C=C (F) C=C4

Molecular Formula

C18H11ClF4N4O3

Molecular Weight

442.75

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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