GRK5-IN-3
GRK5-IN-3 is a potent, covalent small-molecule inhibitor targeting GRK5 and GRK6, with IC50 values of 0.22 μM and 0.41 μM, respectively. This compound is a valuable research tool for investigating GRK5/6 roles in cardiac function, cancer progression, and inflammation through in vitro biochemical and cellular assays.
Product Specifications
CAS Number
2410793-22-3
Field of Research
Cell Biology, Pharmacology & Drug Discovery
Smiles
N (C1=C2C (=NC (NC3=C (OC) C=C (NC (C=C) =O) C=C3) =N1) NC=C2) C4=C (C (N) =O) C=CC=C4
Molecular Formula
C23H21N7O3
Molecular Weight
443.46
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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