BPTF-IN-1
BPTF-IN-1 (AU1) is a selective small-molecule inhibitor of the BPTF bromodomain, demonstrating a Kd of 2.8 μM and greater selectivity over BRD4. This compound exhibits antimalarial activity and serves as a chemical probe for studying chromatin biology and epigenetic mechanisms in both cellular and parasite models.
Product Specifications
CAS Number
2359618-49-6
Field of Research
Epigenetics & Chromatin, Infectious Disease & Virology
Smiles
N (C=1N=C (C=CN1) N2C[C@@H] (NC (NC3=CC (C (OC) =O) =CC=C3) =O) CC2) C4=CC=C (F) C=C4
Molecular Formula
C23H23FN6O3
Molecular Weight
450.47
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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