CPI-1612
CPI-1612 is a potent and orally bioavailable small molecule inhibitor of the EP300/CBP histone acetyltransferase (HAT) activity, with an IC50 of 8.1 nM against EP300 HAT. It demonstrates anticancer properties in research models, facilitating the study of epigenetic mechanisms in oncology and other disease contexts.
Product Specifications
CAS Number
2374971-81-8
Field of Research
Epigenetics & Chromatin
Smiles
C[C@H] (CN[C@@H] (C (=O) Nc1ccc (cn1) -c1cnn (C) c1) c1ccccc1) c1ccc (cc1) C#N
Molecular Formula
C27H26N6O
Molecular Weight
450.53
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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