Aurora A/PKC-IN-1
Aurora A/PKC-IN-1 (Compound 2e) is a potent dual inhibitor of Aurora A and PKC isoforms, demonstrating low nanomolar IC50 values. It exhibits anti-proliferative and anti-metastatic activity in breast cancer cell studies, making it a valuable chemical probe for oncology research, particularly in studying kinase signaling pathways in vitro.
Product Specifications
CAS Number
2143100-98-3
Field of Research
Cell Biology, Epigenetics & Chromatin, Signal Transduction
Smiles
O=C1N ([Se]C=2C1=CC=CC2) C3=NC (NC4CC[Se]C4) =C5C (=N3) N=CN5
Molecular Formula
C16H14N6OSe2
Molecular Weight
464.24
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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