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CDK1-IN-1

CDK1-IN-7 is a potent and selective CDK1/CycB inhibitor (IC50 = 161.2 nM) that induces p53-dependent intrinsic apoptosis. It demonstrates anti-proliferative effects and selective activity in tumor tissue, making it a candidate for targeted cancer therapy research in both cellular and animal models.

Product Specifications

CAS Number

2761858-59-5

Field of Research

Cell Biology

Smiles

C (N) (=O) C1=C2N (C (=CC (=N2) C3=CC=CC=C3) C4=CC=CC=C4) N=C1NC5=C (OC) C=C (OC) C=C5

Molecular Formula

C27H23N5O3

Molecular Weight

465.5

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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