Androgen receptor antagonist 5
This small molecule is a potent androgen receptor (AR) antagonist with an IC50 of 6.17 μM. It demonstrates anti-proliferative activity in LNCaP prostate cancer cells in vitro and exhibits antitumor efficacy in LNCaP xenograft mouse models, making it a valuable tool for prostate cancer research.
Product Specifications
CAS Number
2586195-28-8
Field of Research
Metabolism Research, Pharmacology & Drug Discovery
Smiles
S=C1N2C (C (=O) N1C=3C=C (C (F) (F) F) C (C#N) =NC3) CC=4C (C2) =CC (NC (OCC) =O) =C (F) C4
Molecular Formula
C21H15F4N5O3S
Molecular Weight
493.43
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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