CCG-273220
CCG-273220 is a selective, covalent inhibitor of GRK5 (IC50 220 nM) that targets the subfamily-specific cysteine residue Cys474. It is a valuable research tool for investigating GRK5's role in cardiac function and heart failure models in both cellular and in vivo studies.
Product Specifications
CAS Number
2750414-35-6
Field of Research
Pharmacology & Drug Discovery
Smiles
C[C@@H] (NC (=O) c1ccc2NC (=O) \C (=C/c3[nH]c (C) c (NC (=O) CCl) c3C) c2c1) c1ccc (F) cc1
Molecular Formula
C26H24ClFN4O3
Molecular Weight
494.95
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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