PARP1/BRD4-IN-1
PARP1/BRD4-IN-1 is a potent dual inhibitor of PARP1 (IC50=49 nM) and BRD4 (IC50=202 nM) . It suppresses their expression and activity, demonstrating synergistic anti-proliferative effects in pancreatic cancer cell models in vitro, supporting its use in oncology research.
Product Specifications
CAS Number
2758117-74-5
Field of Research
Cell Biology, Epigenetics & Chromatin, Epigenetics & Chromatin; Cell Biology, Molecular Biology
Smiles
C (N1C (C=2C (N (C) C1=O) =CC=C (C2) C=3C (C) =NOC3C) C4=CC=CC=C4) C=5NC=6C (N5) =CC=CC6C (N) =O
Molecular Formula
C29H26N6O3
Molecular Weight
506.56
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
MBS8431362-02 5x 0.002 mg
Human BMP-5 Recombinant Protein Lyophilized
Sign In for Pricing
View Details 039996-PE 200 µL
PI3KCD, NT (PIK3CD, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform, Phosphatidylinositol 4,5-bisphosphate 3-kinase 110kD catalytic subunit delta) (PE) discontinued
Sign In for Pricing
View Details