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PAD2-IN-1 hydrochloride

PAD2-IN-1 hydrochloride is a benzimidazole-based, potent and selective inhibitor of protein arginine deiminase 2 (PAD2) . It demonstrates high selectivity over PAD4 (95-fold) and PAD3 (79-fold) . This compound is a valuable chemical probe for investigating PAD2 function in rheumatoid arthritis, multiple sclerosis, and other citrullination-related pathologies in cellular and animal models.

Product Specifications

Field of Research

Epigenetics & Chromatin

Molecular Formula

C25H30ClFN6O3

Molecular Weight

517

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

Frequently Asked Questions

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