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XPO1-IN-1

XPO1-IN-1 is an orally bioavailable inhibitor of Exportin 1 (XPO1) with an IC50 of 24 nM in MM.1S multiple myeloma cells. It induces cell cycle arrest and apoptosis in vitro and demonstrates favorable metabolic stability for in vivo pharmacokinetic studies in cancer research.

Product Specifications

Field of Research

Cancer Biology, Cell Biology

Molecular Formula

C20H15F6N5O3S

Molecular Weight

519.42

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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