WDR5-IN-5
WDR5-IN-5 is a potent, selective, and orally bioavailable small molecule inhibitor of the WDR5 WIN site, with sub-nanomolar binding affinity (Ki<0.02 nM) . It demonstrates anti-proliferative activity in cancer cell-based assays and has shown a favorable pharmacokinetic profile in preclinical studies, supporting its use in oncology research.
Product Specifications
CAS Number
2417012-26-9
Field of Research
Epigenetics & Chromatin
Smiles
C (F) (F) (F) C=1C (C2=C3C (C (=O) N ([C@@H] ([C@H]4CC4) C5=CC (C) =CC=N5) CC3) =CC (CN6C=CN=C6) =C2) =CN (CC) N1
Molecular Formula
C29H29F3N6O
Molecular Weight
534.58
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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