ERα antagonist 1
ERα antagonist 1 is a potent and selective covalent inhibitor of estrogen receptor alpha. It induces G0/G1 cell cycle arrest and apoptosis in ERα-positive breast cancer cells like MCF-7, making it a valuable tool for investigating ERα biology and therapeutic strategies in both cellular and animal models of hormone-dependent cancers.
Product Specifications
CAS Number
2762423-09-4
Field of Research
Cell Biology, Metabolism Research, Pharmacology & Drug Discovery
Smiles
C (=O) (C1=C (SC=2C1=CC=C (O) C2) C3=CC=C (O) C=C3) C4=CC=C (OC5CN (C/C=C/C (=O) N6CCCCC6) C5) C=C4
Molecular Formula
C33H32N2O5S
Molecular Weight
568.68
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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