O-Desethyl Dapagliflozin
O-Desethyl Dapagliflozin (Empagliflozin-4) is an active metabolite and potent SGLT2 inhibitor with an IC50 of 33 nM. It is a valuable reference compound for pharmacokinetic and metabolic studies in diabetes research, applicable in both in vitro enzymatic assays and in vivo models.
Product Specifications
CAS Number
864070-37-1
Product Name Alternative
Empagliflozin-4, O-Desethyl Dapagliflozin, SGLT2
Field of Research
Pharmacology & Drug Discovery
Purity
97.09% (May vary between batches)
Solubility
DMSO:27.5 mg/mL (72.21 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:5 mg/mL (13.13 mM)
Smiles
O[C@H]1[C@@H] (O[C@H] (CO) [C@@H] (O) [C@@H]1O) C2=CC (CC3=CC=C (O) C=C3) =C (Cl) C=C2
Molecular Formula
C19H21ClO6
Molecular Weight
380.82
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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