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UNC5293

UNC5293 is a highly potent and selective MERTK inhibitor (Ki = 190 pM) with excellent oral bioavailability. It demonstrates significant selectivity over Axl, Tyro3, and Flt3 and is utilized in leukemia research, particularly for in vivo studies involving bone marrow malignancies.

Product Specifications

CAS Number

2226789-82-6

Field of Research

Cardiovascular Research, Signal Transduction

Smiles

CCC[C@H] (C) Nc1ncc2c (cn ([C@H]3CC[C@H] (O) CC3) c2n1) C1CCN (CC1) C (=O) c1cc (C) nc (C) c1

Molecular Formula

C30H42N6O2

Molecular Weight

518.69

Storage Conditions

-20°C

Notes

For research use only.

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