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APC-6860

APC-6860 is a potent and selective trypsin-like serine protease inhibitor, demonstrating high affinity for urokinase (uPA) with Ki values of 0.1 μM (human) and 0.082 μM (murine) . Its selectivity profile, particularly for uPA over tPA, supports its application in cancer research for studying tumor progression and metastasis in experimental models.

Product Specifications

CAS Number

154628-42-9

Field of Research

Protein Biochemistry

Smiles

NC (=N) c1cc2c (I) cccc2s1

Molecular Formula

C9H7IN2S

Molecular Weight

302.13

Storage Conditions

-20°C

Notes

For research use only.

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