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Haspin-IN-1

Haspin-IN-1 (2a) is a potent, small-molecule inhibitor of haspin kinase (IC50=119 nM) with additional activity against CLK1, DYRK1A, and CDK9. This multi-kinase inhibition profile supports its investigation as a potential anticancer agent in cellular and biochemical research contexts.

Product Specifications

Field of Research

Cell Biology, Epigenetics & Chromatin, Signal Transduction

Molecular Formula

C12H8N4O2S

Molecular Weight

272.28

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

Frequently Asked Questions

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