CXCR2 antagonist 4
CXCR2 antagonist 4 (compound 7) is a potent small molecule inhibitor of the CXCR2 receptor (IC50 = 0.13 μM) and CXCL8-induced calcium mobilization (IC50 = 27 μM) . Its application in cancer research is supported by studies demonstrating its role in inhibiting neutrophil recruitment and tumor progression in preclinical models.
Product Specifications
Field of Research
Cell Biology, Immunology & Inflammation, Immunology & Inflammation; Pharmacology & Drug Discovery, Pharmacology & Drug Discovery
Molecular Formula
C15H14F2N4OS2
Molecular Weight
368.42
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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