P2Y2R/GPR17 antagonist 1
Compound 14m is a dual antagonist targeting both the P2Y2 and GPR17 receptors, exhibiting IC50 values of 3.17 μM and 1.67 μM, respectively. This small molecule is a valuable research tool for investigating purinergic signaling in models of inflammation, neuropathic pain, and demyelinating diseases in vitro.
Product Specifications
CAS Number
2395016-49-4
Product Name Alternative
GPR17
Field of Research
Metabolism Research, Neuroscience, Pharmacology & Drug Discovery
Purity
98.21% (May vary between batches)
Solubility
DMSO:112.5 mg/mL (259.92 mM)
Smiles
[O-][N+] (=O) c1cccc (OS (=O) (=O) c2ccc (NC (=O) c3ccccc3Cl) cc2) c1
Molecular Formula
C19H13ClN2O6S
Molecular Weight
432.83
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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