AT2R antagonist 1
AT2R antagonist 1 is a potent and selective angiotensin II AT2 receptor ligand with a Ki of 29 nM. It exhibits high metabolic stability in human, rat, and mouse liver microsomes but inhibits common CYP enzymes. This profile makes it a valuable pharmacological tool for studying AT2R function in cardiovascular and neurological research models, both in vitro and in vivo.
Product Specifications
CAS Number
2709031-17-2
Field of Research
Metabolism Research, Pharmacology & Drug Discovery
Smiles
S (NC (OC) =O) (=O) (=O) C1=C (N=C (CC (C) C) S1) C2=CC=C (CN3C (C (C) (C) C) =NC=C3) C=C2
Molecular Formula
C23H30N4O4S2
Molecular Weight
490.64
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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