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Hsp90-IN-16

Hsp90-IN-16 is a selective HSP90 inhibitor effective against HER2-positive cancers. It demonstrates potent anti-proliferative activity in HCC1954 breast cancer cells (IC50 = 6 μM) by degrading client proteins like HER2/neu, leading to apoptosis. This compound is a valuable tool for investigating HSP90 biology in oncology research, both in vitro and in vivo.

Product Specifications

Molecular Formula

C30H26FN3O6

Molecular Weight

543.54

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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