EPZ-719
EPZ-719 is a potent and selective small molecule inhibitor of the histone methyltransferase SETD2 (IC50 = 0.005 μM) . Its high selectivity makes it a valuable chemical probe for epigenetic research, enabling the study of SETD2's role in chromatin regulation and disease contexts in both cellular and animal models.
Product Specifications
CAS Number
2697176-16-0
Field of Research
Epigenetics & Chromatin
Purity
99.95% (May vary between batches)
Smiles
FC1=C2C (NC (C (N[C@H]3C[C@H] (CCC3) N4C[C@@H] (N (S (C) (=O) =O) C) CC4) =O) =C2) =C (C) C=C1
Molecular Formula
C22H31FN4O3S
Molecular Weight
450.57
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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