PBRM1-BD2-IN-8
PBRM1-BD2-IN-8 (compound 34) is a selective inhibitor of the PBRM1 bromodomain 2 (BD2), exhibiting potent binding affinity (Kd=4.4 μM) and inhibitory activity (IC50=0.16 μM) . This small molecule demonstrates anti-cancer properties in research settings, enabling the study of chromatin remodeling and gene regulation in both cellular and biochemical assays.
Product Specifications
CAS Number
2819989-75-6
Product Name Alternative
EpigeneticReaderDomain, Epigenetic Reader Domain, PBRM1BD2IN8, PBRM1-BD2-IN-8
Field of Research
Epigenetics & Chromatin
Purity
99.48% (May vary between batches)
Solubility
DMSO:55 mg/mL (173.4 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (6.31 mM)
Smiles
O=C1C=2C (NC (N1) C3=CC (C) =CC=C3) =CC=CC2Br
Molecular Formula
C15H13BrN2O
Molecular Weight
317.18
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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