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NSD1 inhibitor BT5

NSD1 inhibitor BT5 is a covalent, small molecule inhibitor of NSD1 histone methyltransferase with IC50 of 1.4 uM, shows no covalent binding to NSD2.

Product Specifications

CAS Number

2351225-46-0

Field of Research

Epigenetics & Chromatin; Pharmacology & Drug Discovery

Purity

>98%

Smiles

C1C (=CC2SC (N) =NC=2C=1O) N1CC1C

Molecular Formula

C10H11N3OS

Molecular Weight

221.28

Notes

For research use only.

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