VU0152100
VU0152100 is a selective allosteric potentiator of the muscarinic acetylcholine receptor M4, exhibiting an EC50 of 380 nM. This compound is a valuable research tool for investigating M4 receptor function in both in vitro assays and in vivo models related to neuroscience and CNS disorders.
Product Specifications
CAS Number
409351-28-6
Product Name Alternative
Muscarinic acetylcholine receptor, inhibit, mAChR, M4 mAChR, Inhibitor, VU152100, VU-152100, VU 0152100, VU 152100, VU0152100, VU-0152100
Field of Research
Neuroscience
Purity
99.43% (May vary between batches)
Solubility
10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (5.86 mM) ; DMSO:55 mg/mL (161.09 mM)
Smiles
COc1ccc (CNC (=O) c2sc3nc (C) cc (C) c3c2N) cc1
Molecular Formula
C18H19N3O2S
Molecular Weight
341.43
References & Citations
Paulina Cieślik 1, Anna Rafało-Ulińska 1, Joanna M Wierońska Prevention of MK-801-induced amnestic effect with combined activation of 5-HT1A and muscarinic receptors in mice Pharmacol Biochem Behav, (2024)
Pubmed id
38462045
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
