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VU0467154

VU0467154 acts as a positive allosteric modulator selectively targeting the M4 muscarinic acetylcholine receptor. This small molecule is a valuable research tool for investigating M4 receptor function in neuropharmacology, with applications in both in vitro assays and in vivo models for central nervous system disorders.

Product Specifications

CAS Number

1451993-15-9

Product Name Alternative

Inhibitor, Human M4 receptor, inhibit, Muscarinic acetylcholine receptor, mAChR, M4 mAChR, Cynomolgus monkey M4 receptor, Rat M4 receptor, VU0467154, VU-0467154, VU 0467154

Field of Research

Neuroscience

Purity

98.05% (May vary between batches)

Solubility

DMSO:55 mg/mL (123.75 mM)

Smiles

NC=1C=2C (SC1C (NCC3=CC=C (S (C (F) (F) F) (=O) =O) C=C3) =O) =NN=C (C) C2C

Molecular Formula

C17H15F3N4O3S2

Molecular Weight

444.45

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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