Intepirdine
Intepirdine (GSK-742457) is a potent and selective 5-HT6 receptor antagonist investigated for Alzheimer's Disease. It has been utilized in both in vitro binding assays and in vivo cognitive studies in animal models to explore its potential therapeutic effects.
Product Specifications
CAS Number
607742-69-8
Product Name Alternative
5HTReceptor, 5HT Receptor, 5-hydroxytryptamine Receptor, 5-HT6, 5-HT Receptor, inhibit, Inhibitor, GSK742457, GSK-742457, GSK 742457, Intepirdine, SB 742457, SB742457, SB-742457, RVT 101, RVT101, RVT-101, Serotonin Receptor
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Purity
95.19% (May vary between batches)
Solubility
H2O:< 1 mg/mL (insoluble or slightly soluble) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (5.66 mM) ; Ethanol:2 mg/mL (5.66 mM) ; DMSO:70 mg/mL (198.05 mM)
Smiles
S (=O) (=O) (C1=CC2=C (C (=CC=C2) N3CCNCC3) N=C1) C4=CC=CC=C4
Molecular Formula
C19H19N3O2S
Molecular Weight
353.44
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog