GR 103691
GR 103691 is a highly potent and selective dopamine D3 receptor antagonist with a Ki of 0.4 nM, exhibiting over 100-fold selectivity for hD3 over hD4 and hD1 receptors. This compound is a valuable pharmacological tool for investigating D3 receptor function in substance use disorders and Parkinson's disease, applicable in both in vitro binding assays and in vivo behavioral models.
Product Specifications
CAS Number
162408-66-4
Product Name Alternative
Human dopamine D3 receptor, GR-103691, GR103691, GR 103691, Inhibitor, inhibit, D3, DopamineReceptor, Dopamine, Dopamine Receptor
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Purity
98.94% (May vary between batches)
Solubility
DMSO:4.86 mg/mL (10.01 mM)
Smiles
COc1ccccc1N1CCN (CCCCNC (=O) c2ccc (cc2) -c2ccc (cc2) C (C) =O) CC1
Molecular Formula
C30H35N3O3
Molecular Weight
485.62
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
Explore Other Products
Browse additional items from our catalog