EP4 receptor antagonist 1
EP4 Receptor Antagonist 1 is a potent and selective competitive antagonist of the prostanoid EP4 receptor, with IC50 values of 6.1 nM (human) and 16.2 nM (mouse) . It shows >1000-fold selectivity over other EP receptor subtypes. This compound is a valuable research tool for studying EP4's role in cancer immunology and inflammation in both cellular and animal models.
Product Specifications
CAS Number
2287259-07-6
Product Name Alternative
Cancer, cells, Inhibitor, inhibit, immunotherapy, mouse EP4 receptor, EP4 receptor antagonist 1, EP-4 receptor antagonist 1, EP4, HEK293, human EP4 receptor, Prostaglandin Receptor, ProstaglandinReceptor
Field of Research
Immunology & Inflammation, Pharmacology & Drug Discovery
Purity
99.53% (May vary between batches)
Smiles
C\C=C\c1nnn (Cc2ccc (cc2) C (F) (F) F) c1C (=O) N[C@@H] (C) c1ccc (cc1) C (O) =O
Molecular Formula
C23H21F3N4O3
Molecular Weight
458.43
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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