Eplivanserin
Eplivanserin (SR-46349) is a potent and selective 5-HT2A receptor antagonist, exhibiting a Kd of 1.14 nM and an IC50 of 5.8 nM in rat cortical membranes. It is a valuable research tool for studying serotonin signaling in in vitro binding assays and in vivo models related to sleep and psychiatric disorders.
Product Specifications
CAS Number
130579-75-8
Product Name Alternative
Dopamine, 5HTReceptor, 5-hydroxytryptamine Receptor, 5-HT2C, 5-HT2 Receptor, 5-HT2A, 5HT Receptor, 5-HT Receptor, Eplivanserin, Inhibitor, oral, inhibit, Serotonin Receptor, release, SR 46349, SR46349, SR-46349
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Purity
97.04% (May vary between batches)
Solubility
DMSO:50 mg/mL (152.26 mM)
Smiles
CN (C) CCO\N=C (\C=Cc1ccc (O) cc1) c1ccccc1F
Molecular Formula
C19H21FN2O2
Molecular Weight
328.38
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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