MRGPRX1 agonist 1
MRGPRX1 agonist 1 is a potent and selective small molecule activator of the Mas-related G-protein-coupled receptor X1, exhibiting an EC50 of 50 nM. This compound is a valuable research tool for investigating MRGPRX1-mediated signaling in vitro and its role in itch, pain, and allergic responses in preclinical models.
Product Specifications
CAS Number
2377379-39-8
Product Name Alternative
Inhibit, MRGPRX1, MRGPRX1 agonist 1, MRGPRX-1 agonist 1, Inhibitor
Field of Research
Pharmacology & Drug Discovery
Purity
99.59% (May vary between batches)
Solubility
DMSO:125 mg/mL (287.03 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:4 mg/mL (9.18 mM)
Smiles
COc1ccccc1S (=O) (=O) Nc1ccc (C) cc1Oc1ccc2c (N) nccc2c1
Molecular Formula
C23H21N3O4S
Molecular Weight
435.5
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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