PD0176078
PD0176078 is a newly found N-type Calcium channel blocker.
Product Specifications
CAS Number
[248922-46-5]
UNSPSC
12352005
Target
Calcium Channel
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/PD0176078.html
Purity
99.80
Solubility
DMSO : 100 mg/mL (ultrasonic)
Smiles
CC(C)C[C@H](NC)C(NCCCC(C1=CC=C(F)C=C1)C2=CC=C(F)C=C2)=O
Molecular Formula
C23H30F2N2O
Molecular Weight
388.49
References & Citations
[1]TakashiYamamoto, et al. Discovery, structure-activity relationship study, and oral analgesic efficacy of cyproheptadine derivatives possessing N-type calcium channel inhibitory activity. Bioorg Med Chem. 2006 Aug 1;14 (15) :5333-9.|[2]Yamamoto T, et al. Discovery, structure-activity relationship study, and oral analgesic efficacy of cyproheptadine derivatives possessing N-type calcium channel inhibitory activity. Bioorg Med Chem. 2006 Aug 1;14 (15) :5333-9.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
N-type calcium channel
Available Sizes
Curated Selection
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