Astemizole
Astemizole is a long-acting, non-sedative H1 receptor antagonist with minimal anticholinergic activity. It is used in research on allergic conditions like rhinitis and urticaria, and serves as a pharmacological tool in both in vitro binding assays and in vivo models of allergy and asthma.
Product Specifications
CAS Number
68844-77-9
Product Name Alternative
Antihistamine drug, antipruritic, Astemizole, Inhibitor, hERG K+, Laridal, Histamine Receptor, Histaminos, HistamineReceptor, histamine H1-receptor, H1 receptor, inhibit, KcsA, Paralergin, Potassium Channel, R 43512, R-43512, R43512, PotassiumChannel
Field of Research
Immunology & Inflammation, Neuroscience, Pharmacology & Drug Discovery
Purity
>98%
Bioactivity
Herg channel blocker
Form
Powder
Solubility
Soluble in DMSO (up to 25 mg/ml) or in Ethanol (up to 25 mg/ml) .
Smiles
FC1=CC=C (C=C1) CN2C (=NC=3C=CC=CC32) NC4CCN (CCC5=CC=C (OC) C=C5) CC4
Molecular Formula
C28H31FN4O
Molecular Weight
457.6
Storage Conditions
RT
Notes
For research use only.
Other Product Names
1-[ (4-Fluorophenyl) methyl]-N-[1-[2- (4-methoxyphenyl) ethyl]-4-piperidinyl]-1H-benzimidazol-2-amine
Available Sizes
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