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Trilaciclib hydrochloride

Trilaciclib hydrochloride (G1T28 hydrochloride) is a potent and selective CDK4/6 inhibitor with IC50 values of 1 nM and 4 nM for CDK4 and CDK6, respectively. It is widely used in preclinical research to investigate cell cycle arrest, chemoprotection, and antitumor efficacy in both in vitro and in vivo cancer models.

Product Specifications

CAS Number

1977495-97-8

Product Name Alternative

Cyclin dependent kinase, CDK, CDK4/Cyc D1, Cdk4/cyclin D1, cdk6/cyclin D3, CDK6/CyclinD3, Inhibitor, inhibit, G1T28, G1T28 Hydrochloride, G1T28 hydrochloride, Trilaciclib, Trilaciclib hydrochloride, Trilaciclib Hydrochloride

Field of Research

Cell Biology, Pharmacology & Drug Discovery

Purity

98.61% (May vary between batches)

Solubility

DMSO:Insoluble; H2O:10 mM

Smiles

Cl.Cl.CN1CCN (CC1) c1ccc (Nc2ncc3cc4C (=O) NCC5 (CCCCC5) n4c3n2) nc1

Molecular Formula

C24H32Cl2N8O

Molecular Weight

519.47

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

Frequently Asked Questions

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