Elacestrant
Elacestrant is an orally bioavailable selective estrogen receptor degrader (SERD) with preferential activity against ERα (IC50 = 48 nM) over ERβ (IC50 = 870 nM) . It is utilized in research for studying hormone receptor-positive breast cancer, demonstrating antitumor efficacy in both cellular assays and animal models.
Product Specifications
CAS Number
722533-56-4
Product Name Alternative
Estrogen Receptor/ERR, EstrogenReceptor, Estrogen Receptor, Elacestrant, ERβ, ERα, ERR, Inhibitor, inhibit, RAD 1901, RAD-1901, RAD1901, progestogen Receptor, progestogenReceptor
Field of Research
Metabolism Research
Purity
98.31% (May vary between batches)
Solubility
DMSO:60 mg/mL (130.82 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:4 mg/mL (8.72 mM)
Smiles
CCNCCc1ccc (CN (CC) c2cc (OC) ccc2[C@@H]2CCc3cc (O) ccc3C2) cc1
Molecular Formula
C30H38N2O2
Molecular Weight
458.63
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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