Elacestrant dihydrochloride
Elacestrant dihydrochloride is an orally bioavailable selective estrogen receptor degrader (SERD) that demonstrates potent and selective activity against ERα (IC50 = 48 nM) over ERβ. It is utilized in research for studying hormone receptor-positive breast cancer, with applications in both in vitro cellular assays and in vivo xenograft models.
Product Specifications
CAS Number
1349723-93-8
Product Name Alternative
Inhibitor, Elacestrant, Elacestrant Dihydrochloride, Elacestrant dihydrochloride, ERβ, ERα, Estrogen Receptor, EstrogenReceptor, Estrogen Receptor/ERR, inhibit, RAD1901, RAD-1901, RAD1901 Dihydrochloride, RAD1901 dihydrochloride, RAD-1901 Dihydrochloride, RAD 1901 Dihydrochloride, RAD 1901, progestogenReceptor, progestogen Receptor
Field of Research
Metabolism Research
Purity
98.46% (May vary between batches)
Solubility
H2O:40 mg/mL (75.25 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (3.76 mM) ; DMSO:55 mg/mL (103.47 mM)
Smiles
Cl.Cl.CCNCCc1ccc (CN (CC) c2cc (OC) ccc2[C@@H]2CCc3cc (O) ccc3C2) cc1
Molecular Formula
C30H40Cl2N2O2
Molecular Weight
531.56
Storage Conditions
-20°C
Notes
For research use only.
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