CMP8
CMP8 is a selective estrogen receptor ligand with high affinity for mutant ER-LBD, exhibiting IC50 values of 29 nM (MGERα), 41 nM (MGRERα), 1100 nM (hERα), and 2200 nM (hERβ) . This small molecule is a valuable research tool for investigating ER function and selectivity in both cellular and biochemical assays.
Product Specifications
CAS Number
851107-28-3
Product Name Alternative
CMP 8, CMP8, CMP-8, ERR, Estrogen Receptor, EstrogenReceptor, Estrogen Receptor/ERR, Inhibitor, hERα, hERβ, inhibit, MGERα, MGRERα, progestogenReceptor, progestogen Receptor
Field of Research
Metabolism Research
Purity
99.36% (May vary between batches)
Solubility
DMSO:50 mg/mL (94.68 mM)
Smiles
C (C12C (C=3C (C1) =CC (O) =CC3) =C (C (=O) CC2) C4=CC=C (OCCN5CCCCC5) C=C4) C6=CC=C (Cl) C=C6
Molecular Formula
C33H34ClNO3
Molecular Weight
528.08
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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