PROTAC ERRα ligand 1
This compound is a potent and selective ERRα antagonist, with IC50 values of 0.04 μM for ERRα and 2.8 μM for ERRγ. It serves as a key ligand for PROTAC development, enabling the targeted degradation of ERRα for research into its role in cancer, metabolism, and other cellular pathways in vitro.
Product Specifications
CAS Number
1264754-13-3
Product Name Alternative
Inhibitor, ERR, ERRα, ERRγ, Estrogen Receptor, EstrogenReceptor, Estrogen Receptor/ERR, inhibit, progestogen Receptor, progestogenReceptor, PROTAC ERRa ligand 1, PROTAC ERRalpha ligand 1, PROTAC ERRα ligand 1, PROTAC ERRα ligand1, PROTAC ERRα ligand-1
Field of Research
Metabolism Research
Purity
99.02% (May vary between batches)
Solubility
DMSO:120 mg/mL (285.47 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:4 mg/mL (9.52 mM)
Smiles
O (C1=C (C (F) (F) F) C=C (C#N) C=C1) C2=C (OC) C=C (/C=C\3/C (=O) NC (=O) S3) C=C2
Molecular Formula
C19H11F3N2O4S
Molecular Weight
420.36
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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