G-1
G-1 is a nonsteroidal, high-affinity, and selective agonist for GPR30 (GPER), with a Ki value of 11 nM. This compound is employed in both in vitro and in vivo research to study GPER-mediated signaling in fields such as oncology, cardiology, endocrinology, and neuroscience, as documented in scientific literature.
Product Specifications
CAS Number
881639-98-1
Product Name Alternative
ERR, G 1, Estrogen Receptor/ERR, EstrogenReceptor, Estrogen Receptor, GPR30, G1, G-1, inhibit, Inhibitor
Field of Research
Metabolism Research, Pharmacology & Drug Discovery
Purity
98.14% (May vary between batches)
Solubility
DMSO:120 mg/mL (291.06 mM) ; H2O:< 0.1 mg/mL (insoluble) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (4.85 mM)
Smiles
[H][C@@]12CC=C[C@]1 ([H]) c1cc (ccc1N[C@@H]2c1cc2OCOc2cc1Br) C (C) =O
Molecular Formula
C21H18BrNO3
Molecular Weight
412.28
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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