GS-6201
GS-6201 (CVT-6883) is a potent and selective adenosine A2B receptor antagonist with a Ki of 22 nM for the human receptor. This small molecule is a valuable research tool for investigating the role of A2B signaling in areas such as fibrosis, inflammation, and cancer in both cellular and animal models.
Product Specifications
CAS Number
752222-83-6
Product Name Alternative
Human A1 receptors, human A2A receptors, human A2B receptors, human A3 receptors, GS6201, GS-6201, GS 6201, inhibit, Inhibitor, infarction, myocardial, caspase-1, cardiac, CVT 6883, CVT-6883, CVT6883, A2B, acute, airway, affinity, Adenosine Receptor, AdenosineReceptor, selectivity, P1 receptor, reactivity, remodeling
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Purity
98.32% (May vary between batches)
Solubility
10% DMSO+90% Corn Oil:2 mg/mL (4.48 mM) ; DMSO:30 mg/mL (67.2 mM)
Smiles
CCCn1c (=O) n (CC) c2[nH]c (nc2c1=O) -c1cnn (Cc2cccc (c2) C (F) (F) F) c1
Molecular Formula
C21H21F3N6O2
Molecular Weight
446.43
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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