GSK1379725A
GSK1379725A is a potent and selective small molecule ligand for the bromodomain of BPTF, exhibiting a binding affinity (Kd) of 2.8 μM. This compound serves as a valuable chemical probe for investigating the role of BPTF in chromatin remodeling and gene regulation, applicable in both in vitro biochemical and cellular studies.
Product Specifications
CAS Number
1802251-00-8
Product Name Alternative
Inhibit, Inhibitor, Epigenetic Reader Domain, EpigeneticReaderDomain, GSK1379725A, GSK-1379725A, BPTF
Field of Research
Epigenetics & Chromatin
Purity
99.51% (May vary between batches)
Solubility
DMSO:50 mg/mL (111 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (4.44 mM)
Smiles
COC (=O) c1cccc (NC (=O) NC2CCN (C2) c2ccnc (Nc3ccc (F) cc3) n2) c1
Molecular Formula
C23H23FN6O3
Molecular Weight
450.47
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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