BI-671800
BI-671800 is a potent and selective antagonist of the CRTH2 (DP2) receptor, with IC50 values of 4.5 nM (human) and 3.7 nM (mouse) for inhibiting PGD2 binding. This investigational compound is used in research to study allergic asthma mechanisms, supporting both in vitro binding assays and in vivo models of airway inflammation.
Product Specifications
CAS Number
1093108-50-9
Product Name Alternative
AP 761, AP761, AP-761, BI 671800, BI671800, BI-671800, Cmpd A, CRTh2 (DP2) receptor, inhibit, mCRTH2, hCRTH2, Inhibitor, ProstaglandinReceptor, Prostaglandin Receptor
Field of Research
Immunology & Inflammation, Metabolism Research, Pharmacology & Drug Discovery
Purity
98.06% (May vary between batches)
Solubility
DMSO:130 mg/mL (259.22 mM)
Smiles
CN (C) c1nc (Cc2ccc (NC (=O) c3ccc (cc3) C (F) (F) F) cc2) nc (N (C) C) c1CC (O) =O
Molecular Formula
C25H26F3N5O3
Molecular Weight
501.5
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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