BX430
BX430 is a potent, selective, and species-specific noncompetitive allosteric antagonist of human P2X4 receptor channels (IC50 = 0.54 μM) . It serves as a valuable research tool for investigating the role of P2X4 in pathologies such as chronic pain and cardiovascular disease, with utility in both in vitro and in vivo experimental models.
Product Specifications
CAS Number
688309-70-8
Product Name Alternative
P2X Receptor, P2X4, P2XReceptor, P2XRs, receptor, specificity, species, Inhibitor, human P2X4 receptor channels, human, pain, inhibit, Ca channels, BX 430, BX430, BX-430, cardiovascular, Calcium Channel, Ca2+ channels, channels, CalciumChannel, chronic, disease
Field of Research
Metabolism Research, Neuroscience, Pharmacology & Drug Discovery
Purity
97.34% (May vary between batches)
Solubility
DMSO:30 mg/mL (72.62 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (4.84 mM)
Smiles
CC (C) c1cc (Br) c (NC (=O) Nc2cccnc2) c (Br) c1
Molecular Formula
C15H15Br2N3O
Molecular Weight
413.11
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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