CB1 antagonist 2
AM4113 is a potent and selective cannabinoid CB1 receptor antagonist with an in vivo IC50 of 25.5 nM. This compound is a valuable research tool for investigating the endocannabinoid system in studies of metabolism, obesity, and substance abuse, utilizing both in vitro and in vivo experimental models.
Product Specifications
CAS Number
614726-85-1
Product Name Alternative
CannabinoidReceptor, Cannabinoid Receptor, AM 4113, AM-4113, AM4113, CB, CB1, CB1 antagonist 2, CB-1 antagonist 2, Inhibitor, inhibit
Field of Research
Neuroscience; Pharmacology & Drug Discovery, Pharmacology & Drug Discovery
Purity
99.75% (May vary between batches)
Solubility
DMSO:1.9 mg/mL (4.99 mM) ; H2O:< 0.1 mg/mL (insoluble) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:1 mg/mL (2.63 mM)
Smiles
Cc1c (nn (c1-c1ccc (Cl) cc1) -c1ccc (Cl) cc1Cl) C (N) =O
Molecular Formula
C17H12Cl3N3O
Molecular Weight
380.66
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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