Tanzisertib
Tanzisertib (CC-930) is a potent and selective JNK1/2/3 inhibitor with respective IC50 values of 61, 7, and 6 nM. It has demonstrated antifibrotic activity in preclinical research, showing efficacy in both in vitro assays and in vivo models of fibrotic diseases.
Product Specifications
CAS Number
899805-25-5
Product Name Alternative
CC 930, CC930, CC-930, inhibit, JNK3, JNK1, JNK2, JNK, Inhibitor, Tanzisertib
Field of Research
Signal Transduction
Purity
98.66% (May vary between batches)
Solubility
10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (4.46 mM) ; DMSO:33 mg/mL (73.59 mM)
Smiles
N (C=1N (C=2C (N1) =CN=C (N[C@H]3CC[C@H] (O) CC3) N2) [C@H]4CCOC4) C5=C (F) C=C (F) C=C5F
Molecular Formula
C21H23F3N6O2
Molecular Weight
448.44
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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