CCG-63802
CCG-63802 is a reversible, small-molecule inhibitor targeting RGS proteins, specifically disrupting the RGS4-Gα interaction with an IC50 of 1.4 μM. This tool compound is used in vitro to study G protein-coupled receptor (GPCR) signaling pathways and has been applied in research investigating neurological disorders and cardiac function.
Product Specifications
CAS Number
620112-78-9
Product Name Alternative
CCG63802, CCG-63802, CCG 63802, inhibit, inflammation, Inhibitor, reversible, RGS, RGS Protein, RGS19, RGS4, Regulator of G-protein Signaling, Regulators of G-protein Signaling, selective
Field of Research
Pharmacology & Drug Discovery
Purity
90.00% (May vary between batches)
Solubility
DMSO:1.67 mg/mL (3.71 mM)
Smiles
Cc1cccc (Oc2nc3c (C) cccn3c (=O) c2\C=C (/C#N) c2nc3ccccc3s2) c1
Molecular Formula
C26H18N4O2S
Molecular Weight
450.51
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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