CCG-63808
CCG-63808 is a reversible, small-molecule inhibitor targeting RGS proteins, specifically demonstrating potent activity against RGS4 with an IC50 of 1.9 μM in TR-FRET binding assays. This compound is a valuable pharmacological tool for investigating G-protein signaling pathways in both cellular and biochemical research contexts.
Product Specifications
CAS Number
620113-73-7
Product Name Alternative
CCG-63808, CCG63808, CCG 63808, inhibit, Inhibitor, RGS4, RGS Protein, RGS19, Regulator of G-protein Signaling, Regulators of G-protein Signaling
Field of Research
Pharmacology & Drug Discovery
Purity
90.00% (May vary between batches)
Solubility
DMSO:1 mg/mL (2.2 mM)
Smiles
Cc1cccn2c1nc (Oc1ccc (F) cc1) c (\C=C (/C#N) c1nc3ccccc3s1) c2=O
Molecular Formula
C25H15FN4O2S
Molecular Weight
454.48
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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