CGS 15943
CGS 15943 is a potent, orally active non-xanthine adenosine receptor antagonist with high affinity for human A1 (Ki=3.5 nM) and A2A (Ki=4.2 nM) receptors. It is widely used as a pharmacological tool in vitro and in vivo to study adenosine signaling in research areas such as cardiovascular function, neuroprotection, and inflammation.
Product Specifications
CAS Number
104615-18-1
Product Name Alternative
Inhibit, p110δ, p110γ, P1 receptor, Inhibitor, CGS 15943, CGS15943, CGS-15943, AdenosineReceptor, adenosine A2B receptor, adenosine A3 receptor, adenosine A1 receptor, adenosine A2A receptor, Adenosine Receptor, A3, A2A, A2B, A1, Phosphoinositide 3-kinase, PI3K
Field of Research
Neuroscience, Pharmacology & Drug Discovery, Signal Transduction
Purity
97.40% (May vary between batches)
Solubility
DMSO:12.22 mg/mL (42.77 mM) ;10% DMSO+90% Corn Oil:1 mg/mL (3.5 mM)
Smiles
Nc1nc2ccc (Cl) cc2c2nc (nn12) -c1ccco1
Molecular Formula
C13H8ClN5O
Molecular Weight
285.69
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog